托伐普坦中间体，多佐胺中间体

托伐普坦中间体Tolvaptan

1. 7-氯-1,2,3,4-四氢苯并[B]氮杂卓-5-酮 (CAS NO:160129-45-3)

7-Chloro-1,2,3,4-tetrahydrobenzo[b] azepin-5-one

2. 7-氯-1,2,3,4-四氢-1-(2-甲基-4-硝基苯甲酰基)-5H-1-苯并氮杂卓-5-酮

7-Chloro-1,2,3,4-tetrahydro-1-(2-methyl-4-nitrobenzoyl)-5H-1-benzazepine-5-on (CAS NO:137982-91-3)

3. 1-(4-氨基-2-甲基苯甲酰基)-7-氯-1,2,3,4-四氢-5H-1-苯并氮杂卓-5-酮

1-(4-Amino-2-methylbenzoyl)-7-chloro-1,2,3,4-tetrahydro-5H-1-benzazepine-5-one

(CAS NO:137977-97-0)

4. N-[4-[(7-氯-2,3,4,5-四氢-5-氧代-1H-1-苯并氮杂卓-1-基)羰基]-3-甲基苯基]-2-甲基苯甲酰胺

N-[4-[7-Chloro-2,3,4,5-tetrahydro-5-oxo-1H-1-benzazepine-1-yl)carbonyl]-3-methylphenyl]-2-methylbenzamide

(CAS NO:137973-76-3)

多佐胺中间体

1. 多佐胺-2-13-(2-thienylthio)butyric acid  (CAS NO:133359-80-5)

2. 多佐胺-2-2 5,6-dihydro 6- methyl-6H-thieno[2,3-b]thiopyran-2-sulfonamide-4-one

3.  4,5-dihydro-6-methyl-6H-thieno[2,3-b] thiopyran-2-sulfonamide-4-ol 7,7,-dioxide

达泊西汀中间体

1. (R)-(+)-3-氯-1-苯基-1-丙醇3-chloro-1-phenyl-propan-1-ol (CAS NO:100306-33-0)

2. 3-（萘-4氧基）-1-苯基-1-丙醇3-(Naphthalen-4-yloxy)-1-Phenyl propan-1-ol

3. 达泊西汀Dapoxetine (CAS NO:119356-77-3)